BDBM764373 8-(4-fluoro-2,5-dimethylphenyl)-9-(4-((1-(3- fluoropropyl)azetidin-3- ylidene)methyl)phenyl)-6,7-dihydro-5H- benzo[7]annulene-3-carboxylic acid::US20250255848, Example 27

SMILES Cc1cc(C2=C(c3ccc(C=C4CN(CCCF)C4)cc3)c3ccc(C(=O)O)cc3CCC2)c(C)cc1F

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 764373   

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandPNGBDBM764373(8-(4-fluoro-2,5-dimethylphenyl)-9-(4-((1-(3- fluor...)
Affinity DataIC50: 0.5nMAssay Description:MCF7 cells (ATCC) were seeded in 384 wells microplate (collagen coated) at a concentration of 10000 cells/30 μL per well in red phenol free MEM alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent