BDBM764535 US20250257051, Compound 48

SMILES CNC(=O)C1CN(c2ncc(C(N)=O)c(Nc3cccc(-c4ncc(F)cn4)c3OC)n2)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 764535   

TargetNon-receptor tyrosine-protein kinase TYK2 [556-888](Human)
1910 Genetics

US Patent
LigandPNGBDBM764535(US20250257051, Compound 48)
Affinity DataKd:  0.5nMAssay Description:Binding constants for compounds disclosed herein against the JH2 domain are determined by the following protocol for a KINOMEscan® assay (DiscoveRx)....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent