BDBM764861 US20250257062, Compound 45

SMILES C[C@H]1c2c(nn(-c3ccc(F)c4c3CCC4)c2-n2ccn(-c3ccc4c(cnn4C4CC4)c3F)c2=O)CCN1C(=O)c1cc2cc(C3CCOCC3)ccc2n1[C@@]1(c2noc(=O)[nH]2)C[C@@H]1C

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 764861   

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Pharma (China)

US Patent
LigandPNGBDBM764861(US20250257062, Compound 45)
Affinity DataEC50:  0.0150nMAssay Description:1. Cell line and reagent preparation1) Cell line: Flp-In-293-GLP1R2) Medium: DMEM+10% FBS+1×Penicillin-Streptomycin+200 μg/mL HB3) Test buffer: 1×HBS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent