BDBM766186 US20250263426, Compound 139-1

SMILES COC(=O)NCC(C)(C)Nc1nc(N2C[C@@H]3CC(c4ncc5c(n4)CC5)=C[C@@H]3C2)nc2c1[S@](=O)CC2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 766186   

Target3',5'-cyclic-AMP phosphodiesterase 4B2 (PDE4B2)(Human)
Xizang Haisco Pharmaceutical Co.

US Patent
LigandPNGBDBM766186(US20250263426, Compound 139-1)
Affinity DataIC50: 20nMAssay Description:The effect of compounds on PDE4B2 activity was detected using a fluorescence polarization kit (BPS Bioscience, Catalog #60343). According to the inst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/3/2025
Entry Details
US Patent

TargetIsoform 2 of 3',5'-cyclic-AMP phosphodiesterase 4D(Homo sapiens (Human))
Xizang Haisco Pharmaceutical Co.

US Patent
LigandPNGBDBM766186(US20250263426, Compound 139-1)
Affinity DataIC50: 20nMAssay Description:The effect of compounds on PDE4D2 activity was detected using a fluorescence polarization kit (BPS Bioscience, Catalog #60345). During the reaction, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/3/2025
Entry Details
US Patent