BDBM766321 US12398118, Compound C43

SMILES CC(OC(=O)N1CCc2sc(-c3ncc(F)c(Nc4ccc5c(c4)CCNC5=O)n3)cc2C1)C(F)(F)F

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 766321   

TargetRho-associated protein kinase 2(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM766321(US12398118, Compound C43)
Affinity DataIC50: 71nMAssay Description:Before the assay, the following working solutions as needed were formulated with corresponding reagents according to the instruction of the kinase de...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM766321(US12398118, Compound C43)
Affinity DataIC50: 1.00E+4nMAssay Description:Before the assay, the following working solutions as needed were formulated with corresponding reagents according to the instruction of the kinase de...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent