BDBM767440 2-[6-(6-Methylpyridin-2-yl)-5- {thieno[3,2-c]pyridin-2-yl}- 1H,2H,3H-imidazo[1,2- a][1,3]diazol-2-yl]acetic acid::US20250270215, Example 21
SMILES Cc1cccc(-c2nc3n(c2-c2cc4cnccc4s2)CC(CC(=O)O)N3)n1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 767440
Affinity DataIC50: 3nMAssay Description:Briefly, the kinase reaction was performed by incubating 2.6 nM of the purified, commercially available human ALK5 (recombinant TGF β1 N-term GST-tag...More data for this Ligand-Target Pair
