BDBM767454 (3-methyloxetan-3-yl)-4-[3-(2-methoxy-3-pyridyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperazine-1-carboxylate::US20250270222, Compound RC-1

SMILES COC1=NC=CCC1C1C=NN2C=CC(N3CCN(C(=O)OC4(C)COC4)CC3)=NC12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 767454   

TargetBMP-2-inducible protein kinase [38-345,K320A,K321A](Human)
Satellos Bioscience

US Patent
LigandPNGBDBM767454((3-methyloxetan-3-yl)-4-[3-(2-methoxy-3-pyridyl)py...)
Affinity DataIC50: 84.6nMAssay Description:This example describes one illustrative method for determining the IC50 of the compounds of the present invention against BIKE (amino acids S38-E345)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/9/2025
Entry Details
US Patent

TargetCyclin-G-associated kinase [25-335](Human)
Satellos Bioscience

US Patent
LigandPNGBDBM767454((3-methyloxetan-3-yl)-4-[3-(2-methoxy-3-pyridyl)py...)
Affinity DataIC50: 1.05E+3nMAssay Description:This example describes one illustrative method for determining the IC50 of the compounds of the present invention against GAK (amino acids Q25-N335)....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/9/2025
Entry Details
US Patent