BDBM767538 US20250270222, Compound I-86

SMILES CN1C[C@@H](OC(=O)N2CCN(c3ccn4ncc(-c5cc(F)cnc5OC5CC5)c4n3)CC2)CC1=O

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 767538   

TargetBMP-2-inducible protein kinase [38-345,K320A,K321A](Human)
Satellos Bioscience

US Patent
LigandPNGBDBM767538(US20250270222, Compound I-86)
Affinity DataIC50: 325nMAssay Description:This example describes one illustrative method for determining the IC50 of the compounds of the present invention against BIKE (amino acids S38-E345)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/9/2025
Entry Details
US Patent

TargetCyclin-G-associated kinase [25-335](Human)
Satellos Bioscience

US Patent
LigandPNGBDBM767538(US20250270222, Compound I-86)
Affinity DataIC50: 1.50E+3nMAssay Description:This example describes one illustrative method for determining the IC50 of the compounds of the present invention against GAK (amino acids Q25-N335)....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/9/2025
Entry Details
US Patent