BDBM770285 (S)-N-((3S,4S)-1-(imidazo[1,5-a]pyridine-8-carbonyl)-4-phenylpiperidin-3-yl)-3-methyl-2-(methylsulfonamido)butanamide::WO2024107778, Compound 74

SMILES CC(C)[C@H](NS(C)(=O)=O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1

InChI Key InChIKey=OHYBJFDQWUWAPR-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 770285   

TargetReplicase polyprotein 1ab(2019-nCoV)
Takeda Pharmaceutical

WIPO
LigandChemical structure of BindingDB Monomer ID 770285BDBM770285((S)-N-((3S,4S)-1-(imidazo[1,5-a]pyridine-8-carbony...)
Affinity DataIC50: 64.7nMAssay Description: Compounds are 3 fold serially diluted for 10 doses and added to an assay plate (384w format) using ECHO, in duplicate wells. The test concentration ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/25/2025
Entry Details
WIPO WO2024107778

TargetAngiotensin-converting enzyme 2(Human)
Takeda Pharmaceutical

WIPO
LigandChemical structure of BindingDB Monomer ID 770285BDBM770285((S)-N-((3S,4S)-1-(imidazo[1,5-a]pyridine-8-carbony...)
Affinity DataEC50:  7.59E+3nMAssay Description: Compounds are 3 fold serially diluted for 10 doses and added to an assay plate (384w format) using ECHO, in duplicate wells. The test concentration ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/25/2025
Entry Details
WIPO WO2024107778