BDBM770779 4-((S)-1-((S)-1-((6,7-dihydro-[1,4]dioxino[2'',3'':4,5]benzo[1,2-d]thiazol-2-yl)amino)-1-oxopropan-2-yl)-4,4-difluoropiperidin-3-yl)pyridine 1-oxide::WO2025064535, Compound 100
SMILES S1C(=NC2=C1C=C1C(=C2)OCCO1)NC([C@H](C)N1C[C@@H](C(CC1)(F)F)C1=CC=[N+](C=C1)[O-])=O
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 770779
Affinity DataIC50: 17nMAssay Description:FlpIn TRex-MRGPRX2-HEK293 cells (herein TRex-MRPGRX2-HEK) stably transfected to express human MRGPRX2 were maintained at 37oC with 5% CO2 and grown i...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:LAD-2 cells were maintained at 37oC with 5% CO2 and grown in complete StemPro-34 media supplemented with 1% L-Glutamate, 1% penicillin/streptomycin, ...More data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:LAD-2 cells were maintained at 37oC with 5% CO2 and grown in complete StemPro-34 media supplemented with 1% L-Glutamate, 1% penicillin/streptomycin, ...More data for this Ligand-Target Pair