BDBM772404 US12419888, Compound 47

SMILES Cc1ccc2nc(C)cc(C(=O)N3CCC[C@H](c4nnc5ccccn45)C3)c2c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 772404   

TargetProprotein convertase subtilisin/kexin type 9(Human)
Institut De Cardiologie De Montreal

US Patent
LigandPNGBDBM772404(US12419888, Compound 47)
Affinity DataKd:  1.20E+4nMAssay Description:Binding of affinity of SHIM compounds has been determined using surface plasmon spectroscopy on a Biacore T200 (GE Healthcare). Biotinylated PCSK9 (A...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/6/2026
Entry Details
US Patent