BDBM773556 8-(1,3-dimethyl-1H-pyrazol-5-yl)-N-((5-fluoro-2,3-dihydrobenzofuran-4-yl)methyl)-2-methoxypyrido[4,3-d]pyrimidin-5-amine::US12421228, Example 28

SMILES COc1ncc2c(NCc3c(F)ccc4c3CCO4)ncc(-c3cc(C)nn3C)c2n1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 773556   

LigandPNGBDBM773556(8-(1,3-dimethyl-1H-pyrazol-5-yl)-N-((5-fluoro-2,3-...)
Affinity DataIC50: 100nMAssay Description:Table 6: Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each comp...More data for this Ligand-Target Pair
Ligand Info
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Date in BDB:
1/7/2026
Entry Details
US Patent