BDBM773579 8-(1,3-dimethyl-1H-pyrazol-5-yl)-N-((5-fluoro-2,3-dihydrobenzofuran-4-yl)methyl)-2-methoxy-1,6-naphthyridin-5-amine::US12421228, Example 52
SMILES COc5ccc4c(NCc2c(F)ccc1OCCc12)ncc(c3cc(C)nn3C)c4n5
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 773579
TargetHistone-binding protein RBBP4/Histone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2(Human)
Mirati Therapeutics
US Patent
Mirati Therapeutics
US Patent
Affinity DataIC50: 250nMAssay Description:Table 6: Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each comp...More data for this Ligand-Target Pair
Ligand Info
