BDBM773969 4-((1H- pyrazol-1- yl)methyl)-3- ethynyl-N-((6- methoxy-2,3- dihydro-1H- inden-5- yl)sulfonyl) benzamide::US20250304535, Example C9

SMILES C#Cc1cc(C(=O)NS(=O)(=O)c2cc3c(cc2OC)CCC3)ccc1Cn1cccn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 773969   

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandPNGBDBM773969(4-((1H- pyrazol-1- yl)methyl)-3- ethynyl-N-((6- me...)
Affinity DataIC50: 75nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandPNGBDBM773969(4-((1H- pyrazol-1- yl)methyl)-3- ethynyl-N-((6- me...)
Affinity DataIC50: 75nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent