BDBM773978 4-((1H- pyrazol-1- yl)methyl)-3- cyclopropyl- N-((2- methoxy-5-(4- methoxypiperidin- 1- yl)phenyl) sulfonyl) benzamide::US20250304535, Example C17

SMILES COc1ccc(N2CCC(OC)CC2)cc1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(C2CC2)c1

InChI Key InChIKey=RLWPKPNIMKMDTJ-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 773978   

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 773978BDBM773978(4-((1H- pyrazol-1- yl)methyl)-3- cyclopropyl- N-((...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 773978BDBM773978(4-((1H- pyrazol-1- yl)methyl)-3- cyclopropyl- N-((...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent