BDBM773979 4-((1H- pyrazol-1- yl)methyl)-N- ((5-(tert- butyl)-2- methoxyphenyl) sulfonyl)-3- (oxetan-2- yl)benzamide::US20250304535, Example C18

SMILES COc1ccc(C(C)(C)C)cc1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(C2CCO2)c1

InChI Key InChIKey=RBVCAPAUIUUPES-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 773979   

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 773979BDBM773979(4-((1H- pyrazol-1- yl)methyl)-N- ((5-(tert- butyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 773979BDBM773979(4-((1H- pyrazol-1- yl)methyl)-N- ((5-(tert- butyl)...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent