BDBM774015 US12428395, Compound 1.8

SMILES N#Cc1cnc(Nc2cc(NCC3CCNCC3)c(C(F)(F)F)nn2)cn1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 774015   

TargetSerine/threonine-protein kinase Chk1(Human)
Sperogenix Therapeutics

US Patent
LigandPNGBDBM774015(US12428395, Compound 1.8)
Affinity DataIC50: 5.81E+3nMAssay Description:A competitive displacement assay was configured for B-Raf that monitors the amount of a fluorescently-tagged tracer bound to B-Raf via TR-FRET from a...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/14/2026
Entry Details
US Patent