BDBM774133 5-((1H-pyrazol-1- yl)methyl)-6- (methoxy-d3)- N-((6-methoxy-2,2- dimethyl-2,3- dihydrobenzofuran- 7- yl)sulfonyl) picolinamide::US20250304535, Example C65

SMILES [2H]C([2H])([2H])Oc1nc(C(=O)NS(=O)(=O)c2c(OC)ccc3c2OC(C)(C)C3)ccc1Cn1cccn1

InChI Key InChIKey=OWJKOTKNAJAFKP-GKOSEXJESA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 774133   

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774133BDBM774133(5-((1H-pyrazol-1- yl)methyl)-6- (methoxy-d3)- N-((...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774133BDBM774133(5-((1H-pyrazol-1- yl)methyl)-6- (methoxy-d3)- N-((...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent