BDBM774140 5-((1H-pyrazol-1- yl)methyl)- N-((2-(tert- butyl)-5- methoxypyridin-4- yl)sulfonyl)-6- methoxy- picolinamide::US20250304535, Example C72

SMILES COc1cnc(C(C)(C)C)cc1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key InChIKey=LZDVOIUPBZXNIJ-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 774140   

TargetHistone acetyltransferase KAT6A [497-780](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774140BDBM774140(5-((1H-pyrazol-1- yl)methyl)- N-((2-(tert- butyl)-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B [657-1069](Human)
Beigene Switzerland

US Patent
LigandChemical structure of BindingDB Monomer ID 774140BDBM774140(5-((1H-pyrazol-1- yl)methyl)- N-((2-(tert- butyl)-...)
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent