BDBM774720 7-(4-(6-(4- Aminopiperidin-1-yl)- 5-cyano-4-(4-cyano-3- fluorophenyl)-2- methylpyridin-3-yl)-2- hydroxyphenoxy)-N- hydroxyheptanamide hydrochloride::US20250304549, Example 26
SMILES Cc1nc(N2CCC(N)CC2)c(C#N)c(-c2ccc(C#N)c(F)c2)c1-c1ccc(OCCCCCCC(=O)NO)c(O)c1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 774720
Affinity DataIC50: 0.120nMAssay Description:The effect of the compounds on LSD1 enzyme activity was examined using the HTRF technique to assess the level of inhibition. Initially, a master solu...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 35nMAssay Description:The effect of the compound on the enzymatic activity of pan-HDAC and two isoforms (HDAC1 and HDAC8) was examined using the HDAC-Glo I/II Assay and Sc...More data for this Ligand-Target Pair
Ligand Info
