BDBM774980 US20250304563, Compound 134

SMILES C#CCCS(=O)(=O)N1CCN(c2cc(C3(Cc4nncn4C)COC3)cc(N3Cc4c(cc(CN5CCC[C@H](C)C5)cc4C(F)(F)F)C3=O)n2)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 774980   

LigandPNGBDBM774980(US20250304563, Compound 134)
Affinity DataIC50: 12.5nMAssay Description:Compounds were assessed for binding activity to Cbl-b by their ability to compete with and displace a probe comprised of BODIPY-FL fluorophore conjug...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/19/2026
Entry Details
US Patent