BDBM776206 US12435061, Compound 2-143

SMILES Cc1nc(C(=O)N2CCC(c3ccc(-c4ccccc4C4CC4)cc3CO)C2)ccc1O

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 776206   

TargetSodium channel protein type 5 subunit alpha(Human)
Kamari Pharma

US Patent
LigandPNGBDBM776206(US12435061, Compound 2-143)
Affinity DataIC50: 10.3nMAssay Description:Nav1.5 was activated by a voltage step protocol on a Nanion Pathchliner. A cesium fluoride internal solution was used. Normal ringer solution served ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
1/22/2026
Entry Details
US Patent