BDBM788165 US12473303, Compound H-APPAMP-022

SMILES Cc1cccn2cc(CNc3cc(NC[C@H]4CCNC[C@@H]4O)nc4c(C5CC5)cnn34)nc12

InChI Key InChIKey=JKNWTBFFMLNWFL-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 788165   

TargetCyclin-K/Cyclin-dependent kinase 12(Human)
Carrick Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 788165BDBM788165(US12473303, Compound H-APPAMP-022)
Affinity DataIC50: 164nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/8/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 788165BDBM788165(US12473303, Compound H-APPAMP-022)
Affinity DataIC50: 622nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/8/2026
Entry Details
US Patent