BDBM789137 UAMC-000-5036::US20250353833, Inhibitor UAMC0005036

SMILES CC(C)(C)NC(=O)NC12CC3CC(CC(NCC(=O)N4Cc5cc(F)c(F)cc5C4)(C3)C1)C2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 789137   

TargetDipeptidyl peptidase 9(Human)TBA
LigandChemical structure of BindingDB Monomer ID 789137BDBM789137(UAMC-000-5036 | US20250353833, Inhibitor UAMC00050...)
Affinity DataIC50: 0.00600nMAssay Description:Table 3 and 4: IC50 measurements. Enzyme activities were determined kinetically in 96-well half area plates (Greiner Bio-One) in a final volume of 10...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/10/2026
Entry Details

TargetDipeptidyl peptidase 8(Human)TBA
LigandChemical structure of BindingDB Monomer ID 789137BDBM789137(UAMC-000-5036 | US20250353833, Inhibitor UAMC00050...)
Affinity DataIC50: 1.33nMAssay Description:Table 3 and 4: IC50 measurements. Enzyme activities were determined kinetically in 96-well half area plates (Greiner Bio-One) in a final volume of 10...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
3/10/2026
Entry Details