BDBM793870 US20260055108, Compound 47

SMILES CCN(C(=O)c1cc(F)ccc1Oc1nncnc1N1CC2(CCN(CC3CCN(c4ccc(C#N)nn4)CC3)CC2)C1)C(C)C

InChI Key InChIKey=YFMNHEVLDUOURK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 793870   

TargetMenin [2-610](Human)
Hutchmed

US Patent
LigandChemical structure of BindingDB Monomer ID 793870BDBM793870(US20260055108, Compound 47)
Affinity DataIC50: 2.60nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/9/2026
Entry Details
US Patent