BDBM795343 7-[(3-methyl-1H-indazol-6-yl)amino]-2-[2-oxo-2-[2-(trifluoromethyl)morpholin-4-yl]ethyl]isoindolin-1-one::US20260069571, Example 38

SMILES Cc1n[nH]c2cc(Nc3cccc4c3C(=O)N(CC(=O)N3CCOC(C(F)(F)F)C3)C4)ccc12

InChI Key InChIKey=DSFFNADAWSDSIG-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 795343   

TargetEpithelial discoidin domain-containing receptor 1(Human)
Redx Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 795343BDBM795343(7-[(3-methyl-1H-indazol-6-yl)amino]-2-[2-oxo-2-[2-...)
Affinity DataIC50: 10nMAssay Description:Cell-based activity under Prompt Conditions. Rat or human NHE3-mediated Na+-dependent H+ antiport was measured using a modification of the pH sensiti...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/22/2026
Entry Details
US Patent

TargetDiscoidin domain-containing receptor 2(Human)
Redx Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 795343BDBM795343(7-[(3-methyl-1H-indazol-6-yl)amino]-2-[2-oxo-2-[2-...)
Affinity DataIC50: 55nMAssay Description:Cell-based activity under Prompt Conditions. Rat or human NHE3-mediated Na+-dependent H+ antiport was measured using a modification of the pH sensiti...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/22/2026
Entry Details
US Patent