BDBM809023 2-amino-N-{(1S,2S)-2-[(4-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-3,3-dimethyl-2,3-dihydro-1H-indol-5-yl}phenyl)methoxy]cyclopentyl}-5-(prop-1-en-2-yl)pyridine-3-carboxamide::US20260146035, Example 51

SMILES C=C(C)c1cnc(N)c(C(=O)N[C@H]2CCC[C@@H]2OCc2ccc(-c3ccc4c(c3)C(C)(C)CN4C3CCN(CCO)CC3)cc2)c1

InChI Key InChIKey=DNPLHAVBHHHPFB-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 809023   

TargetTyrosine-protein kinase Mer(Human)
Dong-A St Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 809023BDBM809023(2-amino-N-{(1S,2S)-2-[(4-{1-[1-(2-hydroxyethyl)pip...)
Affinity DataIC50: 10nMAssay Description:The reason was carried out in white low volume 384-well plate (Corning, USA) with 25 nL compounds in dimethyl sulfoxide in each well. To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2026
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Dong-A St Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 809023BDBM809023(2-amino-N-{(1S,2S)-2-[(4-{1-[1-(2-hydroxyethyl)pip...)
Affinity DataIC50: 10nMAssay Description:The reason was carried out in white low volume 384-well plate (Corning, USA) with 25 nL compounds in dimethyl sulfoxide in each well. To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2026
Entry Details
US Patent

TargetTyrosinase(Human)
Dong-A St Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 809023BDBM809023(2-amino-N-{(1S,2S)-2-[(4-{1-[1-(2-hydroxyethyl)pip...)
Affinity DataIC50: 10nMAssay Description:The reason was carried out in white low volume 384-well plate (Corning, USA) with 25 nL compounds in dimethyl sulfoxide in each well. To measure the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/14/2026
Entry Details
US Patent