BDBM809032 2-amino-5-(1-methyl-1H-pyrazol-4-yl)-N-[(1S,2S)-2-({4-[1-(propan-2-yl)-1H-indol-5-yl]phenyl}methoxy)cyclopentyl]pyridine-3-carboxamide::US20260146035, Example 60

SMILES CC(C)n1ccc2cc(-c3ccc(CO[C@H]4CCC[C@@H]4NC(=O)c4cc(-c5cnn(C)c5)cnc4N)cc3)ccc21

InChI Key InChIKey=LBLSVYNGRSMQHV-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 809032   

TargetTyrosine-protein kinase Mer(Human)
Dong-A St Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 809032BDBM809032(2-amino-5-(1-methyl-1H-pyrazol-4-yl)-N-[(1S,2S)-2-...)
Affinity DataIC50: 10nMAssay Description:The reason was carried out in white low volume 384-well plate (Corning, USA) with 25 nL compounds in dimethyl sulfoxide in each well. To measure the...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/14/2026
Entry Details
US Patent

TargetTyrosine-protein kinase receptor UFO(Human)
Dong-A St Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 809032BDBM809032(2-amino-5-(1-methyl-1H-pyrazol-4-yl)-N-[(1S,2S)-2-...)
Affinity DataIC50: 55nMAssay Description:The reason was carried out in white low volume 384-well plate (Corning, USA) with 25 nL compounds in dimethyl sulfoxide in each well. To measure the...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/14/2026
Entry Details
US Patent

TargetTyrosinase(Human)
Dong-A St Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 809032BDBM809032(2-amino-5-(1-methyl-1H-pyrazol-4-yl)-N-[(1S,2S)-2-...)
Affinity DataIC50: 1.00E+3nMAssay Description:The reason was carried out in white low volume 384-well plate (Corning, USA) with 25 nL compounds in dimethyl sulfoxide in each well. To measure the...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/14/2026
Entry Details
US Patent