BDBM86751 CHEMBL14935::LY 293558::LY-293558
SMILES OC(=O)[C@@H]1C[C@H]2C[C@@H](CCc3nnn[nH]3)CC[C@H]2CN1
InChI Key InChIKey=ZXFRFPSZAKNPQQ-YTWAJWBKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 22 hits for monomerid = 86751
Affinity DataKi: 2.21E+3nMAssay Description:Inhibition of [3H]-AMPA binding to human Ionontropic glutamate receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity to GluR2More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 2More data for this Ligand-Target Pair
Affinity DataKi: 4.16E+3nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 5More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity to GluR5More data for this Ligand-Target Pair
Affinity DataKi: 9.20E+3nMAssay Description:Binding affinity to GluR1More data for this Ligand-Target Pair
Affinity DataKi: 9.20E+3nMAssay Description:Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 1More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 3More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Binding affinity to GluR3More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 4More data for this Ligand-Target Pair
Affinity DataKi: 5.05E+4nMAssay Description:Binding affinity to GluR4More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Ability to displace binding of [3H]AMPA to recombinant human AMPA receptor Ionotropic glutamate receptor ionotropic kainate 2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Ability to displace binding of [3H]KA to recombinant human KA receptor Ionotropic glutamate receptor ionotropic kainate 2 expressed in EK 293 cell me...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to GluR7More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to GluR6More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-KA binding to iontropic glutamate receptor 6More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of GluK1 receptor (unknown origin)More data for this Ligand-Target Pair