BDBM50529754 CHEMBL579353::GNF-Pf-2789

SMILES CCN(CC)CCCC(C)Nc1nc(\C=C\c2cc(OC)c(OC)cc2Cl)nc2cc(Cl)ccc12

InChI Key InChIKey=ZEHGJPVTWNYYHP-UHFFFAOYSA-N

Data  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50529754   

TargetCalcium/calmodulin-dependent protein kinase type 1G(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of human CAMK1G using KKALRRQETVDAL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1G(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 4.81E+3nMAssay Description:Inhibition of human CAMK1G using KKALRRQETVDAL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 5.15E+3nMAssay Description:Inhibition of human BTK using KVEKIGEGTYGVVYK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 5.15E+3nMAssay Description:Inhibition of human BTK using KVEKIGEGTYGVVYK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase CSK(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 6.85E+3nMAssay Description:Inhibition of human CSK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase CSK(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 6.85E+3nMAssay Description:Inhibition of human CSK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 7.74E+3nMAssay Description:Inhibition of human ERBB4 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 7.74E+3nMAssay Description:Inhibition of human ERBB4 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human LYN-B using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
University of Silesia In Katowice

Curated by ChEMBL
LigandPNGBDBM50529754(CHEMBL579353 | GNF-Pf-2789)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human LYN-B using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed