BDBM50533342 Cebranopadol::GRT-6005::GRT6005
SMILES CN(C)[C@]1(CC[C@@]2(CC1)OCCc1c2[nH]c2ccc(F)cc12)c1ccccc1
InChI Key InChIKey=CSMVOZKEWSOFER-RQNOJGIXSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50533342
Affinity DataKi: 0.700nMAssay Description:Displacement of [N-allyl-2,3-3H]naloxone from recombinant human mu opioid receptor expressed in CHOK1 cell membranes after 90 mins by scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [leucyl-3H]nociceptin from human nociceptin opioid receptor expressed in HEK293 cell membranes after 90 mins by scintillation countin...More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at recombinant human nociceptin opioid receptor expressed in CHOK1 cell membranes after 45 mins by GTPgamma(35)S binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity at recombinant human mu opioid receptor expressed in CHOK1 cell membranes after 45 mins by GTPgamma(35)S binding assayMore data for this Ligand-Target Pair