BDBM50618605 INCB-059872::INCB059872::Incb 59872::Incb-059872

SMILES COCC1(CN[C@@H]2C[C@H]2c2ccccc2)CCN(CC2(CCC2)C(O)=O)CC1

InChI Key InChIKey=WBPWDDPSYSUQJA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50618605   

TargetLysine-specific histone demethylase 1A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50618605(Incb 59872 | Incb-059872 | INCB059872 | INCB-05987...)
Affinity DataIC50: 18nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50618605(Incb 59872 | Incb-059872 | INCB059872 | INCB-05987...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate incubated for 1 hr by fluorescence b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50618605(Incb 59872 | Incb-059872 | INCB059872 | INCB-05987...)
Affinity DataIC50: 18nMAssay Description:Inhibition of N-terminal His-tagged LSD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50618605(Incb 59872 | Incb-059872 | INCB059872 | INCB-05987...)
Affinity DataIC50: 18nMAssay Description:Inhibition of C-terminal His-tagged LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE3) using ART(mK)QTARKSTGGKAPRKQLAGGK-Biotin as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50618605(Incb 59872 | Incb-059872 | INCB059872 | INCB-05987...)
Affinity DataIC50: 18nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed