BDBM50251822 2-(3-ethyl-2-(piperidin-1-yl)-3,4-dihydroquinazolin-4-yl)-N-(4-(4-fluorophenylsulfonamido)benzyl)acetamide::CHEMBL480968::KYS-05065::N-(4-(4-fluorophenylsulfonamido)benzyl)-2-(3-ethyl-2-(piperidin-1-yl)-3,4-dihydroquinazolin-4-yl)acetamide

SMILES CCN1C(CC(=O)NCc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)c2ccccc2N=C1N1CCCCC1

InChI Key InChIKey=PEIFDCMYVCGNKX-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50251822   

TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50251822(N-(4-(4-fluorophenylsulfonamido)benzyl)-2-(3-ethyl...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human T-type calcium channel alpha1G in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50251822(N-(4-(4-fluorophenylsulfonamido)benzyl)-2-(3-ethyl...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of T-type calcium channel Cav3.1 alpha1G expressed in HEK293 cells by whole cell patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed