BDBM50097431 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide::4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide(LUF5433)::4-methoxy-N-(4-phenylthiazol-2-yl)benzamide::CHEMBL60156::LUF-5433

SMILES COc1ccc(cc1)C(=O)Nc1nc(cs1)-c1ccccc1

InChI Key InChIKey=FVWGKRAXWKLEHX-UHFFFAOYSA-N

Data  9 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50097431   

TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortical membrane in presence of 100 uM GTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  670nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  670nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  670nMAssay Description:Displacement of [125I]-AB MECA from human Adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]ZM-241385 from A2A receptor in rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097431(LUF-5433 | 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-ben...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]-CGS-21,680 or [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed