BDBM50494341 LY-293,558::LY-293558::NGX-424::TEZAMPANEL

SMILES [H][C@@]12CC[C@H](CCc3nn[nH]n3)C[C@]1([H])C[C@H](NC2)C(O)=O

InChI Key InChIKey=ZXFRFPSZAKNPQQ-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50494341   

TargetGlutamate receptor 2(Human)
Centro De Investigaci�N Lilly

Curated by ChEMBL
LigandPNGBDBM50494341(LY-293,558 | LY-293558 | NGX-424 | TEZAMPANEL)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 1(Human)
Centro De Investigaci�N Lilly

Curated by ChEMBL
LigandPNGBDBM50494341(LY-293,558 | LY-293558 | NGX-424 | TEZAMPANEL)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed