BDBM50138670 6-Carbamimidoyl-naphthalene-2-carboxylic acid phenylamide::6-[(Z)-AMINO(IMINO)METHYL]-N-PHENYL-2-NAPHTHAMIDE::6-carbamimidoyl-N-phenyl-2-naphthamide::CHEMBL104937::uPa_7
SMILES NC(=N)c1ccc2cc(ccc2c1)C(=O)Nc1ccccc1
InChI Key InChIKey=AECPTICWHONWNW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 29 hits for monomerid = 50138670
Affinity DataKi: 325nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 628nM ΔG°: -8.45kcal/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Inhibition of urokinaseMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Competitive inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins...More data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Inhibition of human plasma plasmin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity towards human plasmin.More data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity value against plasminMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity against plasminMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity value against kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity against human plasma kallikrein.More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity towards P-kallikreinMore data for this Ligand-Target Pair
Affinity DataKi: 5.60E+3nMAssay Description:Binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.64E+3nMAssay Description:Binding affinity against human alpha thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 5.64E+3nMAssay Description:Inhibition of human plasma thrombin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins...More data for this Ligand-Target Pair
Affinity DataKi: 3.18E+4nMAssay Description:Binding affinity value against Tissue plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataKi: 3.18E+4nMAssay Description:Binding affinity towards human Tissue type plasminogen activator.More data for this Ligand-Target Pair
Affinity DataKi: 3.18E+4nMAssay Description:Inhibition of recombinant tPA using H-D-Ile-Pro-Arg-pNA.2HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by sp...More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Binding affinity towards tissue type plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of recombinant tPA using H-D-Ile-Pro-Arg-pNA.2HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by sp...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human plasma plasmin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of human plasma thrombin using pyroGlu-Pro-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins...More data for this Ligand-Target Pair