BDBM1009 N-(3-{1-[4-hydroxy-6,6-bis({[2-(2-methoxyethoxy)ethoxy]methyl})-2-oxo-5,6-dihydro-2H-pyran-3-yl]propyl}phenyl)-1-methyl-1H-imidazole-4-sulfonamide::N-[3-{1-(5,6-Dihydro-4-hydroxy-2-oxo--6,6-bis((2-(2-methoxyethoxy)ethoxy)methyl)-2H-pyran-3-yl)propyl}phenyl]-1-methyl-1H-imidazole-4-sulfonamide::Tipranavir deriv. 21
SMILES CCC(C1C(=O)CC(COCCOCCOC)(COCCOCCOC)OC1=O)c1cccc(NS(=O)(=O)c2cn(C)cn2)c1
InChI Key InChIKey=PXTCOGLXLHGQAQ-UHFFFAOYSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 1009
Affinity DataKi: 28nM ΔG°: -10.2kcal/molepH: 5.0 T: 2°CAssay Description:HIV-1 protease was purified and refolded from E. coli inclusion bodies. The substrate used spans the p17-p24 processing site (R-V-S-Q-N-Y-P-I-V-Q-N-K...More data for this Ligand-Target Pair