BDBM122958 US8735386, IV-9b

SMILES CC1Cc2nn(C)c(Cc3ccccc3Cl)c2-c2nc(Nc3cnn(c3)C3CCN(CC3)C3CCN(CC3)C(C)=O)ncc12

InChI Key InChIKey=QFQNHTDMQSXDJH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 122958   

TargetInsulin-like growth factor 1 receptor(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM122958(US8735386, IV-9b)
Affinity DataIC50: 1nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinase dom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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