BDBM124591 US8759532, 275

SMILES C1CC(CCO1)c1cccnc1Oc1ccc2n(ncc2c1)-c1nc2ccccc2s1

InChI Key InChIKey=MKMSUMXAAHHGHA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 124591   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Amgen

US Patent

LigandBDBM124591(US8759532, 275)Copy SMILESCopy InChI

Affinity DataIC50: 57.9nMT: 2°CAssay Description:To check the inhibition profile, 5 μL of serial diluted compounds were incubated with 5 μL of diluted PDE10 enzyme (BPS Bioscience, San Die...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
11/18/2014
Entry Details
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