BDBM142623 US8933228, 15

SMILES Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ncnc3[nH]c(=O)[nH]c23)c2ccccc12)C(C)(C)C

InChI Key InChIKey=BMKJTSUIIWPPHM-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 142623   

TargetMitogen-activated protein kinase 14(Human)
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US Patent
LigandPNGBDBM142623(US8933228, 15)
Affinity DataIC50: 30nMAssay Description:The enzyme inhibitory activity of test compounds was determined by fluorescence resonance energy transfer (FRET) using synthetic peptides labelled wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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US Patent
LigandPNGBDBM142623(US8933228, 15)
Affinity DataIC50: 35nMAssay Description:The enzyme inhibitory activity of test compounds was determined by fluorescence resonance energy transfer (FRET) using synthetic peptides labelled wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent

TargetTyrosine-protein kinase HCK(Human)
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US Patent
LigandPNGBDBM142623(US8933228, 15)
Affinity DataIC50: 36nMAssay Description:The enzyme inhibitory activity of test compounds was determined by fluorescence resonance energy transfer (FRET) using synthetic peptides labelled wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent

TargetMitogen-activated protein kinase 12(Human)
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US Patent
LigandPNGBDBM142623(US8933228, 15)
Affinity DataIC50: 539nMAssay Description:The enzyme inhibitory activity of test compounds was determined by fluorescence resonance energy transfer (FRET) using synthetic peptides labelled wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
US Patent