BDBM156364 US9018371, 4

SMILES OC1CS[C@H]([C@H]1O)n1cnc2c(NCc3cccc(I)c3)nc(Cl)nc12

InChI Key InChIKey=QMJFSSNSVVHFPD-PMPKIWSKSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 156364   

TargetAdenosine receptor A2a(Homo sapiens (Human))
Fm Therapeutics

US Patent
LigandPNGBDBM156364(US9018371, 4)
Affinity DataKi:  4.16nMAssay Description:CHO cells (ATCC No. CCL-61), in which A1 and A3 adenosine receptors were expressed, were cultured in F-12 media (Gibco, U.S.A.) supplemented with 10%...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Fm Therapeutics

US Patent
LigandPNGBDBM156364(US9018371, 4)
Affinity DataKi:  341nMAssay Description:CHO cells (ATCC No. CCL-61), in which A1 and A3 adenosine receptors were expressed, were cultured in F-12 media (Gibco, U.S.A.) supplemented with 10%...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Fm Therapeutics

US Patent
LigandPNGBDBM156364(US9018371, 4)
Affinity DataKi:  2.49E+3nMAssay Description:CHO cells (ATCC No. CCL-61), in which A1 and A3 adenosine receptors were expressed, were cultured in F-12 media (Gibco, U.S.A.) supplemented with 10%...More data for this Ligand-Target Pair
In DepthDetails US Patent