BDBM176799 US9675612, 36 N-[2-(Dimethylamino)-2-oxoethyl]-7-(1H-indazol-5-ylamino)-N-methyl[1,3]thiazolo[5,4-d]pyrimidine-2-carboxamide

SMILES CN(C)C(=O)CN(C)C(=O)c1nc2c(Nc3ccc4[nH]ncc4c3)ncnc2s1

InChI Key InChIKey=YENCYEMLPGOTLV-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 176799   

TargetIsoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D](Human)
Bayer Pharma Aktiengesellschaft

US Patent

LigandBDBM176799(US9675612, 36 N-[2-(Dimethylamino)-2-oxoethyl]-7-(...)Copy SMILESCopy InChI

Affinity DataIC50: 81nMpH: 7.5Assay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/12/2018
Entry Details
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