BDBM19171 4-phenyl-5H-indeno[1,2-c]pyridazin-5-one::Aza-heterocyclic Derivative, 1i::CHEMBL127880

SMILES O=C1c2ccccc2-c2nncc(c12)-c1ccccc1

InChI Key InChIKey=XXAMPLSBRNFBAB-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 19171   

TargetAmine oxidase [flavin-containing] A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM19171(CHEMBL127880 | 4-phenyl-5H-indeno[1,2-c]pyridazin-...)
Affinity DataIC50: 3.43E+4nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM19171(CHEMBL127880 | 4-phenyl-5H-indeno[1,2-c]pyridazin-...)
Affinity DataIC50: 3.43E+4nMpH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM19171(CHEMBL127880 | 4-phenyl-5H-indeno[1,2-c]pyridazin-...)
Affinity DataIC50: 9.33E+4nMAssay Description:Inhibitory activity against Monoamine oxidase B from rat brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM19171(CHEMBL127880 | 4-phenyl-5H-indeno[1,2-c]pyridazin-...)
Affinity DataIC50: 9.37E+4nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM19171(CHEMBL127880 | 4-phenyl-5H-indeno[1,2-c]pyridazin-...)
Affinity DataIC50: 9.37E+4nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed