BDBM195234 US9670212, 30 3-amino-N-[(8-methyl-2-{methyl[(1-methylpiperidin-3-yl)methyl]amino}quinolin-3-yl)methyl]pyrazine-2-carboxamide

SMILES CN(CC1CCCN(C)C1)c1nc2c(C)cccc2cc1CNC(=O)c1nccnc1N

InChI Key InChIKey=XXYTWHUCYAOSGO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 195234   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Exelixis

US Patent

LigandBDBM195234(US9670212, 30 3-amino-N-[(8-methyl-2-{methyl[(1-me...)Copy SMILESCopy InChI

Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
7/7/2018
Entry Details
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