BDBM212837 US9278960, 1-7::US9636337, 1-7

SMILES Cc1ccc2c(cc(nc2c1)C(N)=O)-c1ccc(F)cc1

InChI Key InChIKey=RTUBBCUPFNQOMU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 212837   

TargetMetabotropic glutamate receptor 2(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM212837(US9278960, 1-7 | US9636337, 1-7)
Affinity DataIC50: 159nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2019
Entry Details
Go to US Patent

LigandPNGBDBM212837(US9278960, 1-7 | US9636337, 1-7)
Affinity DataIC50: 159nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/14/2017
Entry Details
Go to US Patent