BDBM217402 US9212182, 482::US9212182, 483::US9212182, 484

SMILES COc1ccc(cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1)-c1cccc(F)c1

InChI Key InChIKey=WIFFXDVBWBVOHD-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 217402   

LigandPNGBDBM217402(US9212182, 482 | US9212182, 483 | US9212182, 484)
Affinity DataIC50: 54nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2017
Entry Details
US Patent

LigandPNGBDBM217402(US9212182, 482 | US9212182, 483 | US9212182, 484)
Affinity DataIC50: 80nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2017
Entry Details
US Patent

LigandPNGBDBM217402(US9212182, 482 | US9212182, 483 | US9212182, 484)
Affinity DataIC50: 3.23E+4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2017
Entry Details
US Patent