BDBM218114 US9212182, 1145

SMILES COc1cc(C2CC2)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1

InChI Key InChIKey=GCYITIUFGLXGAY-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 218114   

LigandPNGBDBM218114(US9212182, 1145 | US12240839, Compound X)
Affinity DataIC50: 471nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2017
Entry Details
US Patent

LigandPNGBDBM218114(US9212182, 1145 | US12240839, Compound X)
Affinity DataIC50: 48nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent