BDBM226210 US9321790, 22

SMILES FC(F)(F)[C@@H]1CCn2c(nc(cc2=O)N2C[C@@H]3C[C@H]2CO3)N1CC(=O)c1ccc(NC2CC2)nc1

InChI Key InChIKey=JCLAUQZLKAKGKA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 226210   

TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Sanofi

US Patent

LigandBDBM226210(US9321790, 22)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMpH: 7.5Assay Description:The compounds according to the invention underwent pharmacological trials to measure the selectivity toward human lipid kinases and especially human ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/15/2017
Entry Details
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