BDBM247378 US9447095, 9

SMILES Nc1nc(nc(NCc2cncs2)c1Br)-n1ncc2ccccc12

InChI Key InChIKey=YUWMSAPDGLGOKO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 247378   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Palobiofarma

US Patent
LigandPNGBDBM247378(US9447095, 9)
Affinity DataIC50:  1.60nMpH: 7.5Assay Description:The analysis of the activity of the enzyme Phosphodiesterase [3H] cAMP SPA (Perkin Elmer #7090 TRKQ) kit was used for the study of Phosphodiesterase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent