BDBM264060 2-[5-[(4-iodo-2- methoxyphenyl)methoxy]pyrazol- 1-yl]pyridine-4-carboxylic acid::US10173996, Example 145::US9604961, Example 145::US9714230, 145::US9908865, Example 145

SMILES COc1cc(I)ccc1COc1ccnn1-c1cc(ccn1)C(O)=O

InChI Key InChIKey=DNNQPECTYYGIPO-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 264060   

TargetLysine-specific demethylase 5A(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM264060(2-[5-[(4-iodo-2- methoxyphenyl)methoxy]pyrazol- 1-...)
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM264060(2-[5-[(4-iodo-2- methoxyphenyl)methoxy]pyrazol- 1-...)
Affinity DataIC50:  550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetLysine-specific demethylase 5B(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM264060(2-[5-[(4-iodo-2- methoxyphenyl)methoxy]pyrazol- 1-...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent